Cobimetinib；考比替尼；934660-93-2

Formula:C21H21F3IN3O2

Molecular Weight：531.31

Appearance：Off-white solid powder

Purity：98+%

Cobimetinib (GDC-0973, RG7420) is a potent and highly selective MEK1 inhibitor with IC50 of 4.2 nM, and showing no significant inhibition when tested against a panel of more than 100 of serine-threonine and tyrosine kinases. Cobimetinib induces apoptosis. Phase 3.