利那洛肽
Product Name:Linaelotide Acetate
CAS No.:851199-59-2
Synonym:Linzess;Constella
Chemical name:2-(32-amino-40-(2-amino-2-oxoethyl)-26-(2-carboxyethyl)-23-(4-hydroxybenzyl)-9-(1-hydroxyethyl)-3-methyl-1,4,7,10,13,22,25,28,31,38,41,47-dodecaoxotetracontahydro-1H-37,20-(epiminomethano)-6,29-(methanodithiomethano)pyrrolo[2,1-s][1,2,27,28,5,8,11,14,17,20,23,32,35,38,41]tetrathiaundecaazacyclotritetracontine-15-carboxamido)-3-(4-hydroxyphenyl)propanoic acid
Molecular formula:C59H79N15O21S6
Molecular weight:1526.8
Purity(HPLC):≥98%
Biological Activity:
Linaclotide is an peptide agonist of guanylate cyclase 2C that is undergoing clinical trials for use in treating abdominal pain in patients with irritable bowel syndrome (IBS) accompanied by constipation. The drug also has promising outlooks for the treatment of gastroparesis, ulcerative colitis, chronic intestinal pseudo-obstruction (CIPO), and inertia coli as well.
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货号
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CAS No.
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英文名
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C13726
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145781-92-6
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851199-59-2
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120287-85-6(130143-01-0)
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Cetrorelix Acetate
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38916-34-6
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Somatostatin Acetate
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25126-32-3
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Sincalide
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C16939
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196078-30-5
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Pramlintide Acetate
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C13721
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Glucagon Acetate
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C14156
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17034-35-4
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Secretin Acetate
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C13342
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40077-57-4
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Aviptadil Acetate
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C13299
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112568-12-4
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Antide Acetate
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C14062
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24305-27-9
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Protirelin Acetate
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C13296
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20071-00-5
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Angiotensin Acetate
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C13852
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50-57-7
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Lysipressin Acetate
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C13312
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113-79-1
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Argipressin Acetate
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C13607
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60731-46-6
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C13614
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159519-65-0
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69-25-0
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C14246
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103222-11-3
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79561-22-1
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90104-48-6
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107444-51-9
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C16936
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76712-82-8
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