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Etrasimod CAS:1206123-37-6小分子抑制剂
产品型号：C17286
英文简称：
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Product Name:Etrasimod
 
CAS No.:1206123-37-6
 
Synonym:APD-334
 
Chemical name:(R)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid
 
Molecular formula:C26H26F3NO3
 
Molecular weight:457.48
  
Purity(HPLC):98%;ee>99%

Biological Activity:
Etrasimod is a potent, selective and orally available antagonist of the sphingosine-1-phosphate-1 receptor with an IC50 value of 1.88 nM in CHO cells.