现货供应Torin 2
产品型号:C14285
英文简称:
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产品详情
英文名:Torin 2
Chemical Name: 9-(6-Amino-3-pyridinyl)-1-[3-(trifluoromethyl)phenyl]-benzo[h]-1,6-naphthyridin-2(1H)-one
分子式:C24H15F3N4O
分子量:432.40
纯度:>99%
外观:Yellow solid
CAS:1223001-51-1
Biological Activity
Potent and selective mTOR inhibitor (IC50 = 2.1 nM). Displays 800-fold cellular selectivity for mTOR over PI3K (cellular EC50 values are 0.25 and 200 nM for mTOR and PI3K respectively). Orally available.